4-甲基阿米雷司

4-甲基阿米雷司(英语:4-Methylaminorex,缩写4-MAR4-MAX),分子式C10H12N2O,是一种兴奋剂,带有𫫇唑啉基团,由McNeil实验室在1960年代开发[2]

4-甲基阿米雷司
Skeletal formula
Ball-and-stick model of 4-methylaminorex
临床资料
给药途径Oral, Vaporized, Insufflated, Injected
法律规范状态
法律规范
药物动力学数据
生物利用度62% oral; 79% nasal; 91 - 93.5% smoked; 100% IV
药物代谢Hepatic
生物半衰期10-19 hours
排泄途径Renal
识别信息
  • 4-Methyl-5-phenyl-4,5-dihydro-1,3-oxazol-2-amine
CAS号3568-94-3  checkY
29493-77-4  checkY
PubChem CID
DrugBank
ChemSpider
UNII
KEGG
CompTox Dashboard英语CompTox Chemicals Dashboard (EPA)
化学信息
化学式C10H12N2O
摩尔质量176.22 g·mol−1
3D模型(JSmol英语JSmol
手性Racemic mixture
  • CC1C(C2=CC=CC=C2)OC(N)=N1
  • InChI=1S/C10H12N2O/c1-7-9(13-10(11)12-7)8-5-3-2-4-6-8/h2-7,9H,1H3,(H2,11,12) checkY
  • Key:LJQBMYDFWFGESC-UHFFFAOYSA-N checkY

参考文献

  1. ^ Anvisa. RDC Nº 804 - Listas de Substâncias Entorpecentes, Psicotrópicas, Precursoras e Outras sob Controle Especial [Collegiate Board Resolution No. 804 - Lists of Narcotic, Psychotropic, Precursor, and Other Substances under Special Control]. Diário Oficial da União. 2023-07-24 (2023-07-25) [2023-08-27]. (原始内容存档于2023-08-27) (巴西葡萄牙语). 
  2. ^ US 3278382,“2-amino-5-aryloxazoline compositions and methods of using same” 

外部链接